
West Chester, PA 19832 (US)
BROWN, Dean Gordon AstraZeneca
1800 Concord Pike, P.O. Box 15437
Wilmington, DE 19850-5437 (US)
XIAO, Wenhua AstraZeneca
1800 Concord Pike, P.O. Box 15437
Wilmington, DE 19850-5437 (US)
STEELMAN, Gary Banks AstraZeneca
1800 Concord Pike, P.O. Box 15437
Wilmington, DE 19850-5437 (US)
MURPHY, Megan AstraZeneca
1800 Concord Pike, P.O. Box 15437
Wilmington, DE 19850-5437 (US)
HORCHLER, Carey Lynn AstraZeneca
1800 Concord Pike, P.O. Box 15437
Wilmington, DE 19850-5437 (US)
(86)PCT/SE 2000/002607 (en)
(87)WO 2001/047924 5.7.2001
(51) C07 D0477/06 (2006.01)
(11) 01 060 180
(21) 99908540.0
(22)26.02.1999 (86)en
(43)20.12.2000 (87)en
(24) 29.03.2006
(30)02.03.1998 US 76829 P
20.05.1998 GB 9810888
(54) VERFAHREN ZUR SYNTHESE VON
CARBAPENEM-ANTIBIOTIKA
(73)Merck & Co., Inc.
126 East Lincoln Avenue
Rahway, New Jersey 07065 (US)
(72)SKERLJ, Renato
126 East Lincoln Avenue
Rahway, NJ 07065 (US)
HOUGHTON, Peter
126 East Lincoln Avenue
Rahway, NJ 07065 (US)
BRANDS, Karel, M., J.
126 East Lincoln Avenue
Rahway, NJ 07065 (US)
WILLIAMS, John, M.
126 East Lincoln Avenue
Rahway, NJ 07065 (US)
(86)PCT/US 1999/004321 (en)
(87)WO 1999/045010 10.9.1999
(51) C07 D0487/04 (2006.01)
C07 D0487/14 (2006.01)
A61K0031/5517 (2006.01)
A61P0025/18 (2006.01)
(11) 01 377 586
(21) 02731343.6
(22)11.04.2002 (86)en
(43)07.01.2004(87)en
(24) 22.03.2006
(30)12.04.2001 US 283264 P
(54) TRICYCLISCHE DIAZEPINE ALS TOCOLYTISCHE
OXYTOCIN REZEPTOR ANTAGONISTEN
(73)Wyeth
Five Giralda Farms
Madison, New Jersey 07940-0874 (US)
(72)MEMOLI, Kevin, Anthony
The Orchard Apartment 139F
Cranbury, NJ 08512 (US)
FAILLI, Amedeo, Arturo
14 Landing Lane
Princeton Junction, NJ 08550 (US)
SHUMSKY, Jay, Scott
121 Park Avenue
Hightstown, NJ 08520 (US)
CAGGIANO, Thomas, Joseph
350 Stockham Avenue
Morrisville, PA 19067 (US)
SABATUCCI, Joseph, Peter
84 Hunt Club Drive
Collegeville, PA 19426 (US)
TRYBULSKI, Eugene, John
3432 Manor Road
Huntingdon Valley ,PA 19006 (US)
(86)PCT/US 2002/011527 (en)
(87)WO 2002/083678 24.10.2002
(51) C07 D0487/04 (2006.01)
A61K0031/4985 (2006.01)
A61P0003/10 (2006.01)
(11)
01 412 357
(21) 02749813.8
(22)05.07.2002 (86)en
(43)28.04.2004(87)en
(24) 22.03.2006
(30)06.07.2001 US 303474 P
(54) BETA-AMINO-TETRAHYDROIMIDAZO(1,2-A)
PYRAZINE UND -TETRAHYDROTRIAZOLO(4,3-A)
PYRAZINE ALS DIPEPTIDYL PEPTIDASE
INHIBITOREN ZUR BEHANDLUNG ODER
PREVENTION VON DIABETES
(73)Merck & Co., Inc.
126 East Lincoln Avenue
Rahway, New Jersey 07065-0907 (US)
(72)MACCOSS, Malcolm
126 East Lincoln Avenue
Rahway, NJ 07065-0907 (US)
KIM, Dooseop
126 East Lincoln Avenue
Rahway, NJ 07065-0907 (US)
FISHER, Michael, H.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 (US)
PARMEE, Emma, R.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 (US)
WEBER, Ann, E.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 (US)
EDMONDSON, Scott, D.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 (US)
XU, Jinyou
126 East Lincoln Avenue
Rahway, NJ 07065-0907 (US)
(86)PCT/US 2002/021349 (en)
(87)WO 2003/004498 16.1.2003
(51) C07 D0487/04 (2006.01)
(11) 01 436 296
(21) 02774550.4
(22)03.09.2002 (86)en
(43)14.07.2004(87)en
(24) 22.03.2006
(30)11.09.2001 EP 01810875
20.12.2001 EP 01811249
22.03.2002 EP 02405223
(54) VERFAHREN ZUR DIREKTEN HERSTELLUNG VON
PYRROL[3,4-C]PYRROLEN
(73)Ciba Specialty Chemicals Holding Inc.
Klybeckstrasse 141
4057 Basel (CH)
(72)RUFFIEUX, Vincent
Route du Centre 43
1723 Marly (CH)
MODOUX, Florence
Bärenfelserstrasse 3
4057 Basel (CH)
(86)PCT/EP 2002/009791 (en)
(87)WO 2003/022847 20.3.2003
(51) C 07 D 0487/04 (2006.01) Z C 07 D 0231/32 (2006.01)
(11) 01 481 970
(51) C07 D0487/04 (2006.01)
C07 D0209/18 (2006.01)
A61K0031/5025 (2006.01)
(11) 01 492 792
(21) 03730299.9
(22)02.04.2003 (86)fr
(43)05.01.2005(87)fr
(24) 29.03.2006
(30)03.04.2002 FR 0204158
(54) DERIVES DE 3-HETEROARYL-3,5-DIHYDRO-4-OXO-
4H-PYRIDAZINO¬4,5-B|INDOLE-1-ACETAMIDE,LEUR
PREPARATION ET LEUR APPLICATION EN
THERAPEUTIQUE
(73)Sanofi-Aventis
174, Avenue de France
75013 Paris (FR)
(72)FROISSANT, Jacques, Cedex 981
Brevainville
F-41160Morée (FR)
MARABOUT, Benoit
45bis, rue de Versailles
F-91300 Massy (FR)
MARGUET, Frank
17, rue Paul Doumer
F-91370 Verrières Le Buisson (FR)
PUECH, Frédéric
3, allée d’Auvergne
F-78170 La Celle Saint Cloud (FR)
(86)PCT/FR 2003/001027 (fr)
(87)WO 2003/082874 9.10.2003
(51) C07 D0487/06 (2006.01)
C07 D0495/16 (2006.01)
C07 D0491/16 (2006.01)
A61K0031/395 (2006.01)
A61P0025/18 (2006.01)
(11) 01 497 296
(21) 03741766.4
(22)23.04.2003 (86)en
(43)19.01.2005(87)en
(24) 22.03.2006
(30)25.04.2002 US 375349 P
(54) [1,4]DIAZOCINO[7,8,1-hi]INDOLDERIVATE ALS
ANTIPSYCHOTISCHE MITTEL UND MITTEL GEGEN
OBESITÄT
(73)Wyeth
Five Giralda Farms
Madison, New Jersey 07940-0874 (US)
(72)SABB, Annmarie, Louise
15 Meadow Lane
Pennington, NJ 08534 (US)
STACK, Gary, Paul
525 Brookfield Lane
Ambler, PA 19002 (US)
GAO, Hong
24 Reid Avenue
Belle Mead, NJ 08502 (US)
(86)PCT/US 2003/012691 (en)
(87)WO 2003/091257 6.11.2003
(51) C 07 D 0487/14 (2006.01) Z C 07 D 0487/04 (2006.01)
(11) 01 377 586
(51) C 07 D 0487/22 (2006.01) Z A 61 K 0031/409 (2006.01)
(11) 01 404 319
(51) C 07 D 0491/04 (2006.01) Z C 07 D 0231/32 (2006.01)
(11) 01 481 970
(51) C 07 D 0491/10 (2006.01) Z C 07 D 0231/32 (2006.01)
(11)
01 481 970
(51) C 07 D 0491/16 (2006.01) Z C 07 D 0487/06 (2006.01)
(11) 01 497 296
(51) C07 D0493/04 (2006.01)
A61K0031/35 (2006.01)
A61P0019/10 (2006.01)
(11) 01 467 998
(21) 02797167.0
(22)02.12.2002 (86)en
(43)20.10.2004(87)en
(24) 29.03.2006
(30)19.12.2001 US 341957 P
(54) TETRACYCLISCHE HETEROVERBINDUNGEN ALS
MODULATOREN DES ÖSTROGENREZEPTORS
(73)Ortho-McNeil Pharmaceutical, Inc.
U.S. Route No.202
Raritan, NJ 08869-0602 (US)
(72)KANOJIA, Ramesh M., J & J Pharmaceutical R&D
1000 Route 202, Box 300
Raritan, NJ 08869-0602 (US)
JAIN, Nareshkumar F., J & J Pharmaceutical R&D
1000 Route 202, Box 300
Raritan, NJ 08869-0602 (US)
NG, Raymond, J & J Pharmaceutical R&D
1000 Route 202, Box 300
Raritan, NJ 08869-0602 (US)
SUI, Zhihua, J & J Pharmceutical R&D
1000 Route 202, Box 300
Raritan, NJ 08869-0602 (US)
XU, Jiayi, J & J Pharmaceutical R&D
1000 Route 202, Box 300
Raritan, NJ 08869-0602 (US)
(86)PCT/US 2002/038486 (en)
(87)WO 2003/053977 3.7.2003
(51) C07 D0493/10 (2006.01)
(11) 01 366 052
(21) 02715338.6
(22)11.01.2002 (86)en
(43)03.12.2003 (87)en
(24) 22.03.2006
936
+pat+631.3.2006
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